Welcome to our comprehensive guide on male-to-female hormone tablets in feminizing hormone therapy. Male-to-female hormone tablets play a significant role in achieving feminizing effects during the transition journey.
In this article, we will explore the importance of hormone tablets, the different types available, considerations for usage, and provide recommendations for a successful transition.
Let’s embark on this empowering path together.
Understanding Male-to-Female Hormone Tablets: Male-to-female hormone tablets are oral medications prescribed in feminizing hormone therapy to achieve desired feminizing effects.
Medications and Dosage
Anti Androgens
Two anti-androgen options seem to be more widely used than others. These are:
- Cyproterone Acetate at 100mg – 150mg daily, taken orally. This one seems to carry an increased risk of depressive symptoms, and should this side effect occur, the medication is often changed.
- Spironolactone – 100mg- 200mg daily, taken orally. This one might be a good option if you have high blood pressure or are concerned about blood clots or venous thromboembolism as it is a potassium-sparing diuretic.
Other options include:
- Medroxyprogesterone – 5mg – 10mg daily, taken orally, or 150mg monthly via intramuscular injection.
- Nilutamide – 300mg daily, taken orally. This one can cause androgen production in rare cases, so it is usually not the first choice.
- Flutamide – 250mg three times daily, taken orally. This one can also potentially cause androgen production, so it is not the first choice.
Estrogen Treatment
- Ethinyl Estradiol – 100micrograms daily, taken orally. Most effective and easy to come by. It can be in the form of an oral contraceptive pill.
- Conjugated Equine Estrogens – 5mg t- 10mg daily, taken orally. This one is usually not advised as it increases the risk of thrombosis.
- 17ß Estradiol – 2mg – 8mg daily, taken orally, or 200mg monthly intramuscular injection, or 50 – 100micrograms transdermally. This is a synthetic hormone therapy. This option appears to be the most expensive.
- Estriol – 4mg – 6mg daily, taken orally. High doses are necessary for gender affirming hormone therapy.
Here are the important aspects to consider:
- Importance of Hormone Tablets: Hormone tablets are a crucial component of feminizing hormone therapy as they deliver estrogen, progesterone, or a combination of both to help initiate and maintain feminizing changes. These tablets modify hormone levels to align with those typically found in cisgender women, leading to breast development, softer skin, fat redistribution, and other desired feminine characteristics.
- Types of Hormone Tablets: There are various types of hormone tablets used in male-to-female hormone therapy. The most common ones include: (a.) Estrogen Tablets: Estrogen tablets are the primary component of hormone therapy for feminization. They come in different forms, including estradiol, conjugated estrogens, and more. These tablets help elevate estrogen levels and promote feminizing effects. (b.) Progesterone Tablets: Progesterone tablets are sometimes prescribed in addition to estrogen to enhance feminizing effects further and support breast development. Progesterone plays a role in regulating the menstrual cycle and breast tissue development.
- Considerations for Usage: When using male-to-female hormone tablets, it is crucial to consult with a knowledgeable healthcare professional specializing in transgender healthcare. They will assess your needs, overall health, and hormone levels to determine the most suitable hormone tablet regimen. Your healthcare provider will guide you on the proper dosage, potential side effects, and monitoring requirements.
- Dosage and Administration: Hormone tablet dosage and administration vary depending on individual needs and healthcare provider recommendations. It is essential to follow your healthcare provider’s instructions precisely, including the frequency and timing of tablet administration.
- Monitoring and Adjustments: Regular monitoring of hormone levels and follow-up appointments with your healthcare provider are important to ensure the effectiveness of hormone tablets. Hormone levels, liver function, and other relevant parameters will be monitored to optimize your hormone therapy and adjust the dosage if needed.
- Potential Side Effects: Like any medication, hormone tablets may have potential side effects. Common side effects may include breast tenderness, mood changes, bloating, and potential effects on blood clotting. It is important to promptly communicate any concerns or side effects to your healthcare provider. They can guide, make necessary dosage adjustments, or recommend additional measures to mitigate side effects.
Male to Female Hormone Tablets You Can Buy Online
100mg Spironolactone Pills

- SKU:1026
- Generic Brand for Aldactone
- Active Ingredient’s: Spironolactone
- Our Brand: Aldactone
- Strength(mg) :100 mg
- Manufacturer: RPG Life Sciences
- Description: Spironolactone
| PACK SIZE | PRICE PER PILL OR UNIT | PRICE | |
|---|---|---|---|
| 30 Tablet/s | US$0.46 | US$ 13.81 | Add to cart |
| 60 Tablet/s | US$0.46 | US$ 27.63 | Add to cart |
| 90 Tablet/s | US$0.46 | US$ 41.43 | Add to cart |
25mg Spironolactone Pills

- SKU:1305
- Generic Brand for ALDACTONE 25 mg
- Active Ingredient’s: Spironolactone
- Our Brand: ALDACTONE
- Strength(mg) :25mg
- Manufacturer: RPG Life Science
- Description: Aldactone
| PACK SIZE | PRICE PER PILL OR UNIT | PRICE | |
|---|---|---|---|
| 30 Tablet/s | US$0.13 | US$ 3.77 | Add to cart |
| 60 Tablet/s | US$0.13 | US$ 7.54 | Add to cart |
| 90 Tablet/s | US$0.13 | US$ 11.29 | Add to cart |
50mg Androcur Pills
- Sku :290
- Generic Brand for :Androcur
- Active Ingredient’s :Cyproterone Acetate (also spell as Ciproterone Acetate)
- Our Brand :Androcur
- Strength(mg) :50mg
- Manufacturer :Bayer Schering, Turkey
- Description :Cyproterone Acetate (also spell as Ciproterone Acetate)
| PACK SIZE | PRICE PER PILL OR UNIT | PRICE | |
|---|---|---|---|
| 50 Tablet/s | US$1.89 | US$ 94.59 | Add to cart |
| 100 Tablet/s | US$1.89 | US$ 189.19 | Add to cart |
| 150 Tablet/s | US$1.81 | US$ 271.43 | Add to cart |
2mg Estradiol Pills

- SKU:383
- Generic Brand for: Estrace
- Active Ingredient’s: Estradiol
- Our Brand: Progynova
- Strength(mg) :2 mg
- Manufacturer: Zydus Healthcare, India
- Description: Progynova
| PACK SIZE | PRICE PER PILL OR UNIT | PRICE | |
|---|---|---|---|
| 28 Tablet/s | US$0.39 | US$ 11.04 | Add to cart |
| 56 Tablet/s | US$0.39 | US$ 22.07 | Add to cart |
| 84 Tablet/s | US$0.39 | US$ 33.11 | Add to cart |
1mg Estradiol Pills
- SKU:382
- Generic Brand for: Estrace
- Active Ingredient’s: Estradiol
- Our Brand: Progynova
- Strength(mg) :1 mg
- Manufacturer: Zydus Healthcare, India
- Description :
- Expiry :
| PACK SIZE | PRICE PER PILL OR UNIT | PRICE | |
|---|---|---|---|
| 28 Tablet/s | US$0.26 | US$ 7.23 | Add to cart |
| 56 Tablet/s | US$0.26 | US$ 14.46 | Add to cart |
| 84 Tablet/s | US$0.26 | US$ 21.69 | Add to cart |
Climara Forte Estrogen Patches

- Sku :385
- Generic Brand for :Climara Forte
- Active Ingredient’s :Estradiol
- Our Brand :Climara Forte
- Strength(mg) :7.6 mg
- Manufacturer :Bayer Schering Pharma
“Click here to place an order”
| PACK SIZE | PRICE PER PILL OR UNIT | PRICE | |
|---|---|---|---|
| 12 Patches | US$7.61 | US$ 91.35 | |
| 24 Patches | US$7.62 | US$ 182.88 | |
| 36 Patches | US$7.62 | US$ 274.32 |
Conclusion: Male-to-female hormone tablets are an essential component of feminizing hormone therapy, playing a crucial role in achieving desired feminizing effects during the transition journey.
Consultation with a knowledgeable healthcare professional, adherence to the prescribed dosage, regular monitoring, and open communication are vital for a successful hormone therapy experience.
Embrace the transformative power of male-to-female hormone tablets as you navigate this path toward self-discovery, authenticity, and living your true identity.

